SCHEMBL8689665

SCHEMBL8689665

NS(=O)(=O)c1cccc(-n2nc(CO)cc2-c2ccccc2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 16/20 1.00
CA1 P00915 15/20 1.00
CA2 P00918 15/20 1.00
PTGS2 P35354 5/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6344401 0.88 CA9 (1.00) CA9CA1CA2PTGS2
SCHEMBL8689242 0.87 CA1 (0.85) CA9CA1CA2PTGS2
SCHEMBL13239860 0.81 CA1 (0.70) CA9CA1CA2PTGS2
SCHEMBL8033564 0.81 PTGS2 (0.73) CA9CA1CA2PTGS2
SCHEMBL14732172 0.79 CA9 (0.68) CA9CA1CA2PTGS2
Sulfamide SCHEMBL7182772 0.79 PTGS2 (0.76) CA9CA1CA2PTGS2
SCHEMBL3864236 0.78 PTGS2 (0.90) CA9CA1CA2PTGS2
SCHEMBL6406740 0.78 CA9 (0.66) CA9CA1CA2PTGS2
SCHEMBL9941289 0.78 PTGS2 (1.00) CA9CA1CA2PTGS2
SCHEMBL7796498 0.77 CA9 (0.80) CA9CA1CA2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed