SCHEMBL14733989

SCHEMBL14733989

C/C(=C/C(=O)c1ccc(C)c(C)c1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.52
ALDH1A1 P00352 3/20 0.51
CES2 O00748 1/20 0.49
MAOB P27338 2/20 0.48
GAA P10253 1/20 0.46
SRD5A2 P31213 1/20 0.46
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
NR4A1 P22736 1/20 0.44
NR4A2 P43354 1/20 0.44
NR4A3 Q92570 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
HTT P42858 1/20 0.43
RAB9A P51151 1/20 0.43
KCNK3 O14649 1/20 0.42
KCNK9 Q9NPC2 1/20 0.42
POLB P06746 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6703582 0.79 NR4A1 (0.66) S1PR1ALDH1A1CES2MAOBGAA
SCHEMBL6703585 0.79 NR4A1 (0.66) S1PR1ALDH1A1CES2MAOBGAA
SCHEMBL177360 0.79 S1PR1 (0.59) S1PR1ALDH1A1CES2MAOBSRD5A2
SCHEMBL177361 0.79 S1PR1 (0.59) S1PR1ALDH1A1CES2MAOBSRD5A2
SCHEMBL15980075 0.78 CTNNB1 (0.60) ALDH1A1CES2GAASRD5A2MEN1
SCHEMBL7961946 0.77 CES2 (0.57) S1PR1ALDH1A1CES2MAOBGAA
SCHEMBL7961951 0.77 CES2 (0.57) S1PR1ALDH1A1CES2MAOBGAA
SCHEMBL9869192 0.75 ALDH1A1 (0.63) ALDH1A1CES2MAOBSRD5A2MEN1
SCHEMBL7961170 0.75 NPSR1 (0.55) ALDH1A1CES2MAOBGAASRD5A2
SCHEMBL9869199 0.75 ALDH1A1 (0.63) ALDH1A1CES2MAOBSRD5A2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2269993-B1 2-AMINOQUINAZOLINE DERIVATIVE KYOWA HAKKO KIRIN CO LTD (JP) 2013-02-27 EP disclosed