SCHEMBL14735729

SCHEMBL14735729

CC(C)(C)OC(=O)c1ccc2c(C3CCCCC3)c(-c3ccccc3[O])n(C3CCCC3)c2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.39
MMP12 P39900 1/20 0.39
OPRM1 P35372 2/20 0.35
OPRD1 P41143 2/20 0.35
OGFRL1 Q5TC84 2/20 0.35
NR1I2 O75469 3/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
PIM1 P11309 1/20 0.35
MARK3 P27448 1/20 0.35
MAP4K2 Q12851 1/20 0.35
CAMK2B Q13554 1/20 0.35
PIM3 Q86V86 1/20 0.35
PIM2 Q9P1W9 1/20 0.35
SCN9A Q15858 3/20 0.34
KCNH2 Q12809 4/20 0.34
ALDH1A1 P00352 2/20 0.34
ATM Q13315 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1980568 0.91 PRKCA (0.39) PRKCAMMP12OPRM1OPRD1OGFRL1
SCHEMBL1980990 0.85 PTGDR2 (0.41) PRKCAMMP12CYP3A4CYP2C19CYP2D6
SCHEMBL1956510 0.84 PLA2G1B (0.38) PRKCAMMP12OPRM1OPRD1OGFRL1
SCHEMBL1981685 0.82 ALDH1A1 (0.36) OPRM1OPRD1OGFRL1SCN9AALDH1A1
SCHEMBL1980728 0.79 SCN9A (0.42) PRKCAMMP12NR1I2CYP3A4CYP2C19
SCHEMBL2875194 0.78 SCN9A (0.48) PRKCAMMP12NR1I2CYP3A4CYP2C19
SCHEMBL1954406 0.77 PRKCA (0.37) PRKCAMMP12OPRM1OPRD1OGFRL1
SCHEMBL1981129 0.76 PRKCA (0.37) PRKCAMMP12NR1I2CYP3A4CYP2C19
SCHEMBL1956565 0.75 PRKCA (0.48) PRKCAMMP12OGFRL1NR1I2CYP3A4
SCHEMBL752222 0.74 NR1I2 (0.54) PRKCAMMP12NR1I2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2331554-B1 MACROCYCLIC INDOLE DERIVATIVES USEFUL AS HEPATITIS C VIRUS INHIBITORS JANSSEN R & D IRELAND (IE) 2013-03-06 EP disclosed