SCHEMBL14735828

SCHEMBL14735828

COc1ccc(CN2CCN(C)CC2)cc1Nc1ncc(Cl)c(NCc2ccccc2S(N)(=O)=O)n1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 18/20 0.53
INSR P06213 9/20 0.53
AXL P30530 2/20 0.52
AURKA O14965 1/20 0.52
AURKB Q96GD4 1/20 0.52
ROS1 P08922 3/20 0.49
JAK2 O60674 1/20 0.49
SRC P12931 1/20 0.49
TNK2 Q07912 1/20 0.49
MET P08581 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14735829 0.85 ALK (0.54) ALKINSRAXLAURKAAURKB
SCHEMBL375403 0.83 ALK (0.63) ALKINSRAXLAURKAAURKB
SCHEMBL382125 0.78 EGFR (0.69) ALKJAK2SRCTNK2
SCHEMBL5291249 0.74 ALK (0.48) ALKINSRAXLAURKAAURKB
SCHEMBL11916628 0.72 ALK (0.77) ALKINSRAURKAROS1JAK2
SCHEMBL5284485 0.71 ZAP70 (0.45) ALKINSRAXLAURKAAURKB
SCHEMBL1078874 0.71 PRKCQ (0.49) ALKINSRAXLAURKBJAK2
SCHEMBL24255230 0.70 ALK (0.74) ALKINSRAXLJAK2SRC
SCHEMBL6151150 0.70 ZAP70 (0.65) ALK
SCHEMBL20085655 0.70 ALK (0.84) ALKINSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2275413-B1 2,4-di(phenylamino)-pyrimidines useful in the treatment of neoplastic diseases, inflammatory and immune system disorders NOVARTIS AG (CH) 2013-03-06 EP disclosed