SCHEMBL14740689

SCHEMBL14740689

CS(=O)(=O)Nc1ccc(-c2coc3cc(OS(=O)(=O)C(F)(F)F)ccc3c2=O)cc1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH2 P05091 17/20 0.61
STS P08842 1/20 0.55
KDM4E B2RXH2 1/20 0.51
MEN1 O00255 1/20 0.51
NPC1 O15118 1/20 0.51
ALDH1A1 P00352 1/20 0.51
TP53 P04637 1/20 0.51
CYP3A4 P08684 1/20 0.51
MAPT P10636 1/20 0.51
HPGD P15428 1/20 0.51
RAB9A P51151 1/20 0.51
KMT2A Q03164 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
XDH P47989 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18872545 0.88 STS (0.66) ALDH2STSKDM4EMEN1NPC1
SCHEMBL14755355 0.85 ALDH2 (0.58) ALDH2KDM4EMEN1NPC1ALDH1A1
SCHEMBL16372524 0.84 STS (0.76) ALDH2STSKDM4EMEN1NPC1
SCHEMBL14740649 0.84 STS (0.64) ALDH2STSKDM4EMEN1NPC1
SCHEMBL14740635 0.80 STS (0.56) ALDH2STSKDM4EMEN1NPC1
SCHEMBL2107264 0.79 MAOB (0.52) ALDH2ALDH1A1MAPT
SCHEMBL14755324 0.78 ALDH2 (0.71) ALDH2
SCHEMBL17718166 0.78 STS (0.57) ALDH2STSKDM4EMEN1NPC1
SCHEMBL17718161 0.78 STS (0.57) ALDH2STSKDM4EMEN1NPC1
SCHEMBL2107958 0.78 MAOB (0.52) ALDH2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2751090-A1 ALDH-2 INHIBITORS IN THE TREATMENT OF ADDICTION Gilead Sciences, Inc. (US) 2014-07-09 EP disclosed
US-8673966-B2 ALDH-2 inhibitors in the treatment of addiction GILEAD SCIENCES, INC. (US) 2014-03-18 US disclosed
US-20130231325-A1 ALDH-2 INHIBITORS IN THE TREATMENT OF ADDICTION GILEAD SCIENCES. INC. (US) 2013-09-05 US disclosed
WO-2013033377-A1 ALDH-2 INHIBITORS IN THE TREATMENT OF ADDICTION GILEAD SCIENCES, INC. (US) 2013-03-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130231325-A1 ALDH-2 INHIBITORS IN THE TREATMENT OF ADDICTION ALDH1A1, ADH1A, ALDH1B1 ALDH2 5/4885STS 832/4885KDM4E 1604/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.