SCHEMBL14743263

SCHEMBL14743263

CN(C(=O)c1cscn1)c1cc(C(=O)O)cc2cc(Cl)cc(Cl)c12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
ACLY P53396 1/20 0.34
INSR P06213 1/20 0.34
ITK Q08881 1/20 0.34
TPMT P51580 1/20 0.33
PTGES O14684 1/20 0.33
PPM1G O15355 1/20 0.33
ALOX5 P09917 1/20 0.33
PTPN1 P18031 1/20 0.33
KDM5A P29375 1/20 0.33
PPM1A P35813 1/20 0.33
PTPN9 P43378 1/20 0.33
DUSP3 P51452 1/20 0.33
PTPN5 P54829 1/20 0.33
PTPN22 Q9Y2R2 1/20 0.33
GPBAR1 Q8TDU6 3/20 0.32
KDM4A O75164 1/20 0.32
KDM4B O94953 1/20 0.32
KDM5C P41229 1/20 0.32
KDM5B Q9UGL1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14743489 0.84 GAA (0.41) ACLYGPBAR1GRM4NPC1RAB9A
SCHEMBL14743590 0.83 GPBAR1 (0.40) KDM4EGPBAR1ALDH1A1
SCHEMBL14743459 0.82 ACLY (0.36) ACLYTPMTGPBAR1NR1H4NPC1
SCHEMBL14744302 0.81 ACLY (0.46) ACLYTPMTGPBAR1NPC1ALDH1A1
SCHEMBL14743638 0.80 CYP1A2 (0.35) ACLYTPMTGPBAR1GRM4ALDH1A1
SCHEMBL14743375 0.80 GPBAR1 (0.39) ACLYGPBAR1GRM4
SCHEMBL14743703 0.80 ACLY (0.35) ACLYGPBAR1NR1H4NPC1ALDH1A1
SCHEMBL14743723 0.79 KDM4E (0.47) KDM4EACLYGPBAR1GRM1
SCHEMBL14743805 0.76 GPBAR1 (0.43) KDM4EGPBAR1NPC1ALDH1A1HTT
SCHEMBL14743833 0.72 MAPT (0.38) ACLYALOX5NPC1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013030358-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2013-03-07 WO disclosed