SCHEMBL14743459

SCHEMBL14743459

CN(C(=O)c1ncccn1)c1cc(C(=O)O)cc2cc(Cl)cc(Cl)c12

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACLY P53396 1/20 0.36
GPBAR1 Q8TDU6 8/20 0.36
TPMT P51580 1/20 0.35
TP53 P04637 1/20 0.35
NR1H4 Q96RI1 1/20 0.33
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32
MDM2 Q00987 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GPR55 Q9Y2T6 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
AURKA O14965 1/20 0.32
KMO O15229 1/20 0.32
HCAR1 Q9BXC0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14743988 0.87 HTT (0.39) ACLYGPBAR1NPC1ALDH1A1MAPT
SCHEMBL14743489 0.87 GAA (0.41) ACLYGPBAR1TP53NPC1RAB9A
SCHEMBL14743723 0.84 KDM4E (0.47) ACLYGPBAR1
SCHEMBL14743590 0.84 GPBAR1 (0.40) GPBAR1ALDH1A1
SCHEMBL14744302 0.84 ACLY (0.46) ACLYGPBAR1TPMTTP53NPC1
SCHEMBL14743375 0.83 GPBAR1 (0.39) ACLYGPBAR1
SCHEMBL14743638 0.83 CYP1A2 (0.35) ACLYGPBAR1TPMTALDH1A1MAPT
SCHEMBL14743263 0.82 KDM4E (0.38) ACLYGPBAR1TPMTNR1H4NPC1
SCHEMBL14743805 0.81 GPBAR1 (0.43) GPBAR1NPC1ALDH1A1HTTRAB9A
SCHEMBL14743703 0.81 ACLY (0.35) ACLYGPBAR1NR1H4NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013030358-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2013-03-07 WO disclosed