SCHEMBL14743271

SCHEMBL14743271

COc1ccc(NC(=O)C[S@@+]([O-])c2cccc(C)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
HPGD P15428 1/20 0.49
DRD4 P21917 1/20 0.48
RAB9A P51151 3/20 0.48
NPC1 O15118 3/20 0.48
TP53 P04637 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
NFKB1 P19838 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
ALDH1A1 P00352 3/20 0.47
MAPT P10636 1/20 0.47
MTNR1A P48039 2/20 0.46
MTNR1B P49286 2/20 0.46
HTT P42858 1/20 0.46
CRHBP P24387 1/20 0.46
CRHR2 Q13324 1/20 0.46
KCNK3 O14649 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14744393 1.00 MEN1 (0.49) MEN1KMT2AHPGDDRD4RAB9A
SCHEMBL14743269 1.00 MEN1 (0.49) MEN1KMT2AHPGDDRD4RAB9A
SCHEMBL14743287 0.90 MTNR1B (0.54) MEN1KMT2AHPGDRAB9ANPC1
SCHEMBL14743109 0.87 CYP1A2 (0.48) MEN1KMT2AHPGDRAB9ANPC1
SCHEMBL14743108 0.87 CYP1A2 (0.48) MEN1KMT2AHPGDRAB9ANPC1
SCHEMBL14743319 0.87 CYP1A2 (0.48) MEN1KMT2AHPGDRAB9ANPC1
SCHEMBL14743130 0.86 TSHR (0.50) MEN1KMT2AHPGDRAB9ANPC1
SCHEMBL14743445 0.83 NPC1 (0.54) MEN1KMT2ARAB9ANPC1TP53
SCHEMBL14743997 0.81 ALDH1A1 (0.50) MEN1KMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL14743203 0.80 KMT2A (0.53) MEN1KMT2ARAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2758370-A1 PARP INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2014-07-30 EP claimed
WO-2013030205-A1 PARP INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2013-03-07 WO claimed
EP-2758370-A1 PARP INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2014-07-30 EP disclosed
WO-2013030205-A1 PARP INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2013-03-07 WO disclosed