SCHEMBL14744328

SCHEMBL14744328

O=[N+]([O-])c1ccc(-c2ccccc2OC(F)(F)F)c(-c2ccncc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 5/20 0.52
CYP11B1 P15538 5/20 0.52
CYP11B2 P19099 5/20 0.52
PTPRC P08575 3/20 0.45
S100A4 P26447 2/20 0.45
BCHE P06276 1/20 0.45
ACHE P22303 1/20 0.45
CES1 P23141 1/20 0.45
GCGR P47871 1/20 0.41
MAPK14 Q16539 1/20 0.41
MAPT P10636 2/20 0.41
HSP90AA1 P07900 1/20 0.41
CDK5 Q00535 1/20 0.41
CDK5R1 Q15078 1/20 0.41
NCOA1 Q15788 1/20 0.41
NCOA3 Q9Y6Q9 1/20 0.41
PTGS2 P35354 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14746841 0.90 PTGS2 (0.50) CYP19A1CYP11B1CYP11B2PTPRCS100A4
SCHEMBL14746632 0.87 CYP11B1 (0.54) CYP19A1CYP11B1CYP11B2PTPRCS100A4
SCHEMBL14744533 0.87 RORC (0.49) CYP19A1CYP11B1CYP11B2PTPRCS100A4
SCHEMBL14747059 0.85 CYP19A1 (0.40) CYP19A1CYP11B1CYP11B2PTPRCS100A4
SCHEMBL14743965 0.83 PTPRC (0.42) CYP19A1CYP11B1CYP11B2PTPRCS100A4
SCHEMBL14746823 0.82 PTPRC (0.44) CYP19A1CYP11B1CYP11B2PTPRCS100A4
SCHEMBL14744512 0.81 RORC (0.50) CYP19A1PTPRCS100A4BCHEACHE
SCHEMBL14746840 0.81 PTPRC (0.40) CYP19A1CYP11B1CYP11B2PTPRCS100A4
SCHEMBL14744310 0.81 PTPRC (0.42) CYP19A1CYP11B1CYP11B2PTPRCS100A4
SCHEMBL14746814 0.80 RORC (0.52) PTPRCS100A4BCHEACHECES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013029338-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2013-03-07 WO disclosed