SCHEMBL14744310

SCHEMBL14744310

O=[N+]([O-])c1ccc(-c2ccccc2OC(F)(F)F)c(-c2cccnn2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRC P08575 3/20 0.42
S100A4 P26447 2/20 0.42
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42
CES1 P23141 1/20 0.42
MAPT P10636 3/20 0.39
TDP1 Q9NUW8 2/20 0.39
HSP90AA1 P07900 1/20 0.39
CDK5 Q00535 1/20 0.39
CDK5R1 Q15078 1/20 0.39
NCOA1 Q15788 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.39
BAX Q07812 2/20 0.37
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14746823 0.86 PTPRC (0.44) PTPRCS100A4BCHEACHECES1
SCHEMBL14744328 0.81 CYP19A1 (0.52) PTPRCS100A4BCHEACHECES1
SCHEMBL14746632 0.80 CYP11B1 (0.54) PTPRCS100A4BCHEACHECES1
SCHEMBL14746841 0.80 PTGS2 (0.50) PTPRCS100A4BCHEACHECES1
SCHEMBL14744238 0.80 PTPRC (0.40) PTPRCS100A4BCHEACHECES1
SCHEMBL14746789 0.79 PTPRC (0.39) PTPRCS100A4BCHEACHECES1
SCHEMBL14744512 0.79 RORC (0.50) PTPRCS100A4BCHEACHECES1
SCHEMBL14744533 0.77 RORC (0.49) PTPRCS100A4BCHEACHECES1
SCHEMBL14744240 0.77 HSPB1 (0.47) PTPRCS100A4BCHEACHECES1
SCHEMBL14746568 0.77 SCN10A (0.45) PTPRCS100A4BCHEACHECES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013029338-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2013-03-07 WO disclosed