SCHEMBL14744456

SCHEMBL14744456

Cc1cc(-c2cc(N)ccc2-c2ccccc2OC(F)(F)F)ccn1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 1/20 0.45
FEN1 P39748 1/20 0.45
CYP2C9 P11712 3/20 0.44
CYP2D6 P10635 2/20 0.44
KCNH2 Q12809 1/20 0.44
GPR142 Q7Z601 1/20 0.44
SCN9A Q15858 13/20 0.44
PDK2 Q15119 1/20 0.43
S1PR1 P21453 3/20 0.40
TRPA1 O75762 1/20 0.39
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31729824 0.87 GRM2 (0.41) CYP2C9CYP2D6KCNH2GPR142SCN9A
SCHEMBL14744477 0.83 ALOX5AP (0.46) ALOX5APFEN1SCN9AS1PR1TRPA1
SCHEMBL14744308 0.79 ALOX5AP (0.45) ALOX5APFEN1SCN9AS1PR1TRPA1
SCHEMBL14743932 0.78 RORC (0.48) ALOX5APFEN1SCN9AS1PR1TRPA1
SCHEMBL14746755 0.75 RORC (0.54) ALOX5APFEN1SCN9APDK2
SCHEMBL14744102 0.74 RORC (0.49) ALOX5APFEN1CYP2C9SCN9AS1PR1
SCHEMBL14746770 0.74 SCN10A (0.50) ALOX5APFEN1SCN9AS1PR1
SCHEMBL31729829 0.72 GLA (0.43) PDK2S1PR1
SCHEMBL24032682 0.71 POLB (0.62) ALOX5APFEN1SCN9APDK2S1PR1
SCHEMBL1492639 0.71 DYRK1A (0.49) CYP2C9CYP2D6S1PR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013029338-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2013-03-07 WO disclosed