SCHEMBL14744102

SCHEMBL14744102

Nc1ccc(-c2ccccc2OC(F)(F)F)c(-c2ccno2)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.49
CYP1A2 P05177 1/20 0.41
CYP19A1 P11511 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
S1PR1 P21453 5/20 0.40
ALOX5AP P20292 1/20 0.40
FEN1 P39748 1/20 0.40
SCN10A Q9Y5Y9 2/20 0.39
SCN9A Q15858 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
ALDH1A1 P00352 2/20 0.37
ADRA1A P35348 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
ADRA1D P25100 1/20 0.37
ADRA1B P35368 1/20 0.37
KCNN4 O15554 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14744512 0.80 RORC (0.50) RORCCYP1A2CYP19A1CYP2C9CYP2C19
SCHEMBL14746770 0.77 SCN10A (0.50) S1PR1ALOX5APFEN1SCN10ASCN9A
SCHEMBL14743932 0.75 RORC (0.48) RORCS1PR1ALOX5APFEN1SCN10A
SCHEMBL14744456 0.74 ALOX5AP (0.45) CYP2C9S1PR1ALOX5APFEN1SCN9A
SCHEMBL14744206 0.74 PLA2G7 (0.45) RORCALOX5APFEN1SCN10ASCN9A
SCHEMBL24032682 0.74 POLB (0.62) RORCS1PR1ALOX5APFEN1SCN10A
SCHEMBL14744245 0.74 RORC (0.45) RORCALOX5APFEN1SCN10ASCN9A
SCHEMBL30321020 0.74 RORC (0.45) RORCALOX5APFEN1SCN10ASCN9A
SCHEMBL30320923 0.74 POLB (0.62) RORCS1PR1ALOX5APFEN1SCN10A
SCHEMBL14744477 0.73 ALOX5AP (0.46) RORCS1PR1ALOX5APFEN1SCN10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013029338-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2013-03-07 WO disclosed