SCHEMBL14745397

SCHEMBL14745397

C=Cc1c(C=O)cc2ccn(C)c2c1F

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.37
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14745727 0.80 CYP2A6 (0.38) CYP2A6KDM4EALDH1A1
SCHEMBL14745903 0.70 CYP2A6 (0.51) CYP2A6KDM4EALDH1A1MAPT
SCHEMBL18697197 0.68 CYP2A6 (0.53) CYP2A6KDM4EALDH1A1
SCHEMBL2312217 0.68 CYP2A6 (0.41) CYP2A6KDM4EALDH1A1
SCHEMBL9779072 0.68 ALDH1A1 (0.39) CYP2A6KDM4EALDH1A1MEN1KMT2A
SCHEMBL21135077 0.67 PTGS2 (0.34) CYP2A6
SCHEMBL18876145 0.66 CDK4 (0.38) CYP2A6KDM4E
SCHEMBL690926 0.65 CYP2A6 (0.41) CYP2A6KDM4EALDH1A1MEN1KMT2A
SCHEMBL29935861 0.65 CYP2A6 (0.41) CYP2A6KDM4EALDH1A1MEN1KMT2A
SCHEMBL18912153 0.65 CYP2A6 (0.41) CYP2A6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2750678-B1 ANTIBACTERIAL COMPOUNDS AND METHODS FOR USE PTC THERAPEUTICS INC (US) 2017-03-22 EP disclosed
US-20150038438-A1 ANTIBACTERIAL COMPOUNDS AND METHODS FOR USE PTC THERAPEUTICS, INC. 2015-02-05 US disclosed
EP-2750678-A1 ANTIBACTERIAL COMPOUNDS AND METHODS FOR USE PTC Therapeutics, Inc. (US) 2014-07-09 EP disclosed
WO-2013033228-A1 ANTIBACTERIAL COMPOUNDS AND METHODS FOR USE PTC THERAPEUTICS, INC. (US) 2013-03-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150038438-A1 ANTIBACTERIAL COMPOUNDS AND METHODS FOR USE MRPL21, SLC11A2, CLPP CYP2A6 3494/4885KDM4E 4305/4885ALDH1A1 3792/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.