SCHEMBL14748445

SCHEMBL14748445

CC(C)(C)OC(=O)COc1cc(Oc2ccc3c(c2)COB3)ccc1C#N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 6/20 0.44
RAB9A P51151 4/20 0.37
NPC1 O15118 3/20 0.37
HSD17B10 Q99714 3/20 0.37
TP53 P04637 2/20 0.37
AR P10275 1/20 0.36
HPGD P15428 4/20 0.35
POLB P06746 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
MAPT P10636 2/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
PDE4A P27815 2/20 0.34
PDE4C Q08493 2/20 0.34
PDE4D Q08499 2/20 0.34
FFAR1 O14842 1/20 0.34
ALDH1A1 P00352 5/20 0.34
KDM4E B2RXH2 4/20 0.34
TSHR P16473 2/20 0.34
MEN1 O00255 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14748463 0.88 PDE4B (0.47) PDE4BRAB9ANPC1HSD17B10TP53
SCHEMBL14748461 0.85 TBXA2R (0.36) PDE4BARMAPTPDE4APDE4C
SCHEMBL8007244 0.84 PDE4B (0.42) PDE4BRAB9ANPC1HSD17B10TP53
SCHEMBL19622210 0.83 PDE4B (0.44) PDE4BRAB9ANPC1HSD17B10TP53
SCHEMBL2531250 0.80 PDE4B (0.68) PDE4BPDE4APDE4CPDE4D
SCHEMBL14748447 0.79 HPGD (0.42) PDE4BHSD17B10TP53HPGDPOLB
SCHEMBL14748366 0.79 PDE4B (0.42) PDE4BARPDE4APDE4CPDE4D
SCHEMBL19622201 0.79 PDE4B (0.48) PDE4BARPOLBPDE4APDE4C
SCHEMBL19622212 0.78 PDE4B (0.53) PDE4BPDE4APDE4CPDE4D
SCHEMBL13515779 0.77 NPC1 (0.58) RAB9ANPC1HSD17B10TP53AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2564857-A1 Boron-containing small molecules as anti-inflammatory agents Anacor Pharmaceuticals, Inc. (US) 2013-03-06 EP disclosed