SCHEMBL19622201

SCHEMBL19622201

COCCOc1cc(Oc2ccc3c(c2)COB3)ccc1C#N

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 10/20 0.48
AR P10275 5/20 0.43
PDE4A P27815 4/20 0.35
PDE4C Q08493 3/20 0.35
PDE4D Q08499 3/20 0.35
CYP19A1 P11511 1/20 0.34
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
RAF1 P04049 1/20 0.32
MAP2K1 Q02750 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14748463 0.80 PDE4B (0.47) PDE4BARPDE4APDE4CPDE4D
SCHEMBL19622210 0.79 PDE4B (0.44) PDE4BARPDE4APDE4CPDE4D
SCHEMBL14748445 0.79 PDE4B (0.44) PDE4BARPDE4APDE4CPDE4D
SCHEMBL14748366 0.79 PDE4B (0.42) PDE4BARPDE4APDE4CPDE4D
SCHEMBL8007244 0.78 PDE4B (0.42) PDE4BARPDE4APDE4CPDE4D
SCHEMBL14748444 0.77 AR (0.39) PDE4BARPDE4APDE4CPDE4D
SCHEMBL2529313 0.77 PDE4B (0.81) PDE4BPDE4APDE4CPDE4D
SCHEMBL7997145 0.77 AR (0.45) PDE4BARPDE4APDE4CPDE4D
SCHEMBL8004927 0.77 PDE4B (0.56) PDE4BARPDE4APDE4CPDE4D
SCHEMBL14748450 0.77 PDE4B (0.44) PDE4BARPDE4APDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246034-A1 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS Anacor Pharmaceuticals, Inc. (US) 2017-11-22 EP disclosed