SCHEMBL14748447

SCHEMBL14748447

CC1CCN(C(=O)COc2cc(Oc3ccc4c(c3)COB4)ccc2C#N)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.42
ALDH1A1 P00352 6/20 0.41
MAPT P10636 3/20 0.41
KDM4E B2RXH2 3/20 0.41
HSD17B10 Q99714 3/20 0.41
KMT2A Q03164 2/20 0.41
GAA P10253 2/20 0.41
TSHR P16473 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
PDE4B Q07343 2/20 0.41
L3MBTL1 Q9Y468 3/20 0.40
MEN1 O00255 1/20 0.40
SCN7A Q01118 2/20 0.39
KCNH2 Q12809 2/20 0.39
LMNA P02545 3/20 0.39
MAPK1 P28482 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
ESR1 P03372 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2533228 0.82 PDE4B (0.64) PDE4B
SCHEMBL14748463 0.80 PDE4B (0.47) HPGDALDH1A1MAPTKDM4EHSD17B10
SCHEMBL19622210 0.80 PDE4B (0.44) ALDH1A1HSD17B10PDE4BTP53
SCHEMBL14748445 0.79 PDE4B (0.44) HPGDALDH1A1MAPTKDM4EHSD17B10
SCHEMBL8007244 0.78 PDE4B (0.42) HPGDALDH1A1HSD17B10TSHRPDE4B
SCHEMBL19622201 0.76 PDE4B (0.48) GAAPDE4BPOLB
SCHEMBL14748366 0.74 PDE4B (0.42) PDE4BKCNH2
SCHEMBL14748444 0.72 AR (0.39) PDE4BKCNH2
SCHEMBL8007185 0.72 PDE4B (0.67) PDE4BSCN7AKCNH2
SCHEMBL14748448 0.71 PDE4B (0.41) PDE4BPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246034-A1 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS Anacor Pharmaceuticals, Inc. (US) 2017-11-22 EP disclosed
EP-2564857-A1 Boron-containing small molecules as anti-inflammatory agents Anacor Pharmaceuticals, Inc. (US) 2013-03-06 EP disclosed