SCHEMBL14758258

SCHEMBL14758258

Bc1ccc2nc(CO)cn2c1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.42
KDM4E B2RXH2 5/20 0.39
TP53 P04637 2/20 0.39
RAB9A P51151 9/20 0.39
NPC1 O15118 8/20 0.39
SMN1; SMN2 Q16637 5/20 0.39
POLB P06746 2/20 0.39
ALDH1A1 P00352 4/20 0.37
MAPT P10636 2/20 0.37
RXFP1 Q9HBX9 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PKM P14618 2/20 0.35
CYP2C19 P33261 1/20 0.35
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12669969 0.86 KDM4E (0.37) MCHR1KDM4ETP53RAB9ANPC1
SCHEMBL870522 0.79 NPC1 (0.50) MCHR1KDM4ETP53RAB9ANPC1
SCHEMBL9598573 0.78 PIK3CG (0.55) MCHR1KDM4ETP53RAB9ANPC1
SCHEMBL9598420 0.78 KDM4E (0.63) KDM4ETP53RAB9ANPC1SMN1; SMN2
SCHEMBL871183 0.78 GRM5 (0.47) MCHR1KDM4ETP53RAB9ANPC1
SCHEMBL973963 0.78 DRD2 (0.43) MCHR1KDM4ETP53RAB9ANPC1
SCHEMBL9597339 0.73 MCHR1 (0.50) MCHR1KDM4ETP53RAB9ANPC1
SCHEMBL21355035 0.73 METTL3 (0.47) MCHR1
SCHEMBL19292088 0.73 MCHR1 (0.39) MCHR1KDM4ETP53RAB9ANPC1
SCHEMBL102061 0.72 KDM4E (0.56) KDM4ETP53RAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013033258-A1 ANTIBACTERIAL COMPOUNDS AND METHODS FOR USE PTC THERAPEUTICS, INC. (US) 2013-03-07 WO disclosed