SCHEMBL14764213

SCHEMBL14764213

CCc1ccc(O)c([O])c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.64
DAO P14920 2/20 0.49
POLB P06746 1/20 0.49
BACE1 P56817 1/20 0.46
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
ALDH1A1 P00352 3/20 0.41
MAPT P10636 2/20 0.41
KDM4E B2RXH2 1/20 0.41
USP2 O75604 1/20 0.41
GAA P10253 1/20 0.41
ALOX15 P16050 1/20 0.41
ALOX12 P18054 1/20 0.41
HTT P42858 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ESR1 P03372 2/20 0.40
ESR2 Q92731 2/20 0.40
IAPP P10997 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2A6 P11509 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14764389 0.82 TRPA1 (0.64) TRPA1DAOPOLBBACE1ALDH1A1
SCHEMBL1021944 0.79 BACE1 (0.68) TRPA1DAOPOLBBACE1CNR1
SCHEMBL56556 0.78 TRPA1 (1.00) TRPA1POLBBACE1CNR1ALDH1A1
SCHEMBL30290839 0.78 TRPA1 (1.00) TRPA1POLBBACE1CNR1ALDH1A1
SCHEMBL14764068 0.77 ABAT (0.46) TRPA1POLBBACE1ALDH1A1MAPT
SCHEMBL29763176 0.76 TRPA1 (0.70) TRPA1DAOPOLBBACE1CNR1
SCHEMBL2862097 0.76 TRPA1 (0.44) TRPA1DAOPOLBBACE1ALDH1A1
SCHEMBL8047684 0.76 TRPA1 (0.70) TRPA1DAOPOLBBACE1CNR1
Bicarbonate SCHEMBL8911264 0.76 TRPA1 (0.83) TRPA1POLBCNR1ALDH1A1MAPT
SCHEMBL4818051 0.74 TRPA1 (0.43) TRPA1ALDH1A1MAPTKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190085007-A1 4-methylcatechol Derivatives and Uses Thereof Thanares GmbH (DE) 2019-03-21 US claimed
US-20160347782-A1 4-methylcatechol Derivatives and Uses Thereof Thanares GmbH (DE) 2016-12-01 US claimed
WO-2013034119-A1 4-METHYLCATECHOL DERIVATIVES UND USE THEREOF Thanares GmbH (DE) 2013-03-14 WO claimed
US-20190085007-A1 4-methylcatechol Derivatives and Uses Thereof Thanares GmbH (DE) 2019-03-21 US disclosed
US-20160347782-A1 4-methylcatechol Derivatives and Uses Thereof Thanares GmbH (DE) 2016-12-01 US disclosed
WO-2013034119-A1 4-METHYLCATECHOL DERIVATIVES UND USE THEREOF Thanares GmbH (DE) 2013-03-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190085007-A1 4-methylcatechol Derivatives and Uses Thereof ST3GAL3, GALE, DPP4 TRPA1 3958/4885DAO 1794/4885POLB 4824/4885
US-20160347782-A1 4-methylcatechol Derivatives and Uses Thereof ST3GAL3, GALE, DPP4 TRPA1 3958/4885DAO 1794/4885POLB 4824/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.