SCHEMBL14764266

SCHEMBL14764266

C1=Cc2occ3c4ccccc4nc-3c2NC1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BCHE P06276 4/20 0.36
ACHE P22303 3/20 0.36
NQO2 P16083 1/20 0.33
NISCH Q9Y2I1 1/20 0.32
ELANE P08246 3/20 0.31
KDM4E B2RXH2 2/20 0.31
USP2 O75604 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
RXFP1 Q9HBX9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4514403 0.71 KDM4E (0.41) ACHENQO2NISCHKDM4EUSP2
SCHEMBL4488123 0.69 ACHE (0.37) BCHEACHEKDM4EALDH1A1MAPT
SCHEMBL14310463 0.60
SCHEMBL9857769 0.60 ALDH1A1 (0.41) ACHENQO2KDM4EALDH1A1MAPT
SCHEMBL7544635 0.59 PLAUR (0.35) BCHEACHENQO2ELANEKDM4E
SCHEMBL10514970 0.58 PLAUR (0.51) ELANEKDM4EALDH1A1MAPTHPGD
SCHEMBL4507436 0.57 MAPT (0.50) ELANEKDM4EUSP2ALDH1A1MAPT
SCHEMBL11242361 0.57 KDM4E (0.39) ACHEELANEKDM4EUSP2ALDH1A1
SCHEMBL6293469 0.57
SCHEMBL11247647 0.57 GPR3 (0.41) BCHEACHEELANEKDM4EUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013033971-A1 TETRACYCLIC HETEROCYCLE COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEASES MERCK SHARP & DOHME CORP. (US) 2013-03-14 WO disclosed