SCHEMBL14764993

SCHEMBL14764993

COc1ccc2c(c1)NC(=O)C(C)N2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRPF1 P55201 1/20 0.56
CREBBP Q92793 1/20 0.56
ALDH1A1 P00352 2/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
PTPN1 P18031 1/20 0.44
TP53 P04637 1/20 0.43
PDE3B Q13370 2/20 0.43
PDE3A Q14432 2/20 0.43
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
SNCA P37840 1/20 0.42
CA2 P00918 2/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA4 P22748 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
KDM4E B2RXH2 1/20 0.41
GLA P06280 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29160849 0.78 TP53 (0.49) ALDH1A1MEN1KMT2ATP53PDE3B
SCHEMBL24853337 0.78 TP53 (0.49) ALDH1A1MEN1KMT2ATP53PDE3B
SCHEMBL7174583 0.77 BRPF1 (0.52) BRPF1CREBBPALDH1A1MEN1KMT2A
SCHEMBL14765191 0.77 CREBBP (0.61) BRPF1CREBBPALDH1A1MEN1KMT2A
SCHEMBL11654866 0.76 PDE3B (0.47) CREBBPALDH1A1PDE3BPDE3AMAOA
SCHEMBL16053338 0.76 BRPF1 (0.59) BRPF1CREBBPMEN1KMT2ATP53
SCHEMBL2136049 0.76 BRPF1 (0.59) BRPF1CREBBPMEN1KMT2ACA2
SCHEMBL21606298 0.75 MEN1 (0.60) BRPF1CREBBPALDH1A1MEN1KMT2A
SCHEMBL30908507 0.75 MEN1 (0.60) BRPF1CREBBPALDH1A1MEN1KMT2A
SCHEMBL4848196 0.75 CA2 (0.47) ALDH1A1TP53PDE3BPDE3AMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013034755-A1 TRIAZOLOPYRAZINE DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed