SCHEMBL14765152

SCHEMBL14765152

Cc1nc2cc(F)ccc2[nH]c1=O

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 14/20 0.53
KDM4E B2RXH2 1/20 0.52
DAO P14920 1/20 0.47
CASP3 P42574 1/20 0.45
TYMS P04818 1/20 0.44
KEAP1 Q14145 1/20 0.44
NFE2L2 Q16236 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2178282 0.86 KDM4E (0.52) BRD4KDM4EDAOCASP3TYMS
SCHEMBL14765197 0.82 MAPT (0.56) BRD4KDM4EDAO
SCHEMBL6304037 0.79 HRH4 (0.56) BRD4KDM4EDAOTYMS
SCHEMBL14474327 0.79 CASP3 (0.45) BRD4CASP3TYMS
SCHEMBL31180759 0.79 KDM4E (0.62) BRD4KDM4EDAOTYMS
SCHEMBL6304503 0.79 KDM4E (0.44) BRD4KDM4E
SCHEMBL2008567 0.78 TYMS (0.49) KDM4ETYMSKEAP1NFE2L2
SCHEMBL29778147 0.77 KDM4E (0.49) BRD4KDM4EDAOTYMS
SCHEMBL30695515 0.77 ALDH1A1 (0.58) BRD4KDM4ETYMS
SCHEMBL707140 0.77 ALDH1A1 (0.58) BRD4KDM4ETYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023104148-A1 SMALL MOLECULE PROBE BINDING TO α-SYNUCLEIN AGGREGATE AND APPLICATION THEREOF 复旦大学 2023-06-15 WO disclosed
WO-2014139983-A1 [1,2,4]TRIAZOLO[4,3-A]QUINOXALINES AS DUAL PDE2/PDE10 INHIBITORS H. LUNDBECK A/S (DK) 2014-09-18 WO disclosed
WO-2013034755-A1 TRIAZOLOPYRAZINE DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed