SCHEMBL14765285

SCHEMBL14765285

O=C1C(O)=C(CC=CBr)C(=O)c2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APAF1 O14727 3/20 0.50
TDP2 O95551 3/20 0.50
MAPT P10636 6/20 0.47
MEN1 O00255 5/20 0.47
KMT2A Q03164 5/20 0.47
DHODH Q02127 4/20 0.47
KDM4E B2RXH2 4/20 0.47
ALDH1A1 P00352 3/20 0.47
CDC25B P30305 3/20 0.47
CDC25A P30304 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
CYP3A4 P08684 2/20 0.47
TP53 P04637 1/20 0.47
PKM P14618 1/20 0.47
RPS6KA3 P51812 1/20 0.47
GLO1 Q04760 1/20 0.47
GPR35 Q9HC97 1/20 0.47
P2RX7 Q99572 3/20 0.42
MAPK1 P28482 4/20 0.40
CYP1A2 P05177 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6052720 0.83 MAPT (0.51) APAF1TDP2MAPTMEN1KMT2A
SCHEMBL5821364 0.79 APAF1 (0.65) APAF1TDP2MAPTMEN1KMT2A
SCHEMBL939989 0.79 APAF1 (0.54) APAF1TDP2MAPTMEN1KMT2A
SCHEMBL8462690 0.78 MAPT (0.47) APAF1TDP2MAPTMEN1KMT2A
SCHEMBL12127298 0.76 DHODH (0.79) APAF1TDP2MAPTMEN1KMT2A
Lapachol SCHEMBL31492698 0.76 DHODH (0.79) APAF1TDP2MAPTMEN1KMT2A
Lapachol SCHEMBL157255 0.76 DHODH (0.79) APAF1TDP2MAPTMEN1KMT2A
SCHEMBL1520566 0.75 APAF1 (0.65) APAF1TDP2MAPTMEN1KMT2A
Lapachol SCHEMBL18769814 0.75 DHODH (0.77) APAF1TDP2MAPTMEN1KMT2A
Lapachol SCHEMBL3274147 0.75 DHODH (0.77) APAF1TDP2MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013036766-A1 SMALL MOLECULE NAPHTHOQUINONE- AND PHTHALIMIDE-BASED LIPOCATIONS AS ANTI-PARASITIC AGENTS UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 2013-03-14 WO disclosed