SCHEMBL14767409

SCHEMBL14767409

Nc1ccc(-c2ccc(COc3ccc(CN4CCCC4)cc3)nc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 15/20 0.55
ALDH1A1 P00352 1/20 0.52
HRH4 Q9H3N8 1/20 0.48
TSHR P16473 1/20 0.45
ACHE P22303 1/20 0.45
RAD52 P43351 1/20 0.45
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12440662 0.89 HRH3 (0.57) HRH3ALDH1A1HRH4CYP2D6
SCHEMBL12441461 0.76 MCHR1 (0.57) HRH3HRH4TSHR
SCHEMBL19291552 0.75 HRH3 (0.62) HRH3HRH4CYP2D6CYP2C19
SCHEMBL54966 0.73 ALDH1A1 (0.96) HRH3ALDH1A1HRH4CYP2D6CYP2C19
SCHEMBL31010237 0.73 HRH3 (0.66) HRH3TSHRACHERAD52
SCHEMBL12440536 0.72 KDM4E (0.55) HRH3ALDH1A1HRH4CYP2D6CYP2C19
SCHEMBL62541 0.72 ALDH1A1 (1.00) HRH3ALDH1A1HRH4CYP2D6CYP2C19
SCHEMBL10616916 0.72 ALDH1A1 (1.00) HRH3ALDH1A1HRH4CYP2D6CYP2C19
SCHEMBL3156543 0.72 ALDH1A1 (1.00) HRH3ALDH1A1HRH4CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL5521932 0.72 ALDH1A1 (0.92) HRH3ALDH1A1HRH4ACHECYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558578-B1 NOVEL ALKYNE COMPOUNDS HAVING AN MCH ANTAGONISTIC EFFECT AND MEDICAMENTS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM PHARMA (DE) 2013-03-13 EP disclosed