SCHEMBL14767428

SCHEMBL14767428

Nc1ccc(-c2ccc(-c3ccc(NCCN4CCCC4)cc3)nc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.54
ADRA2A P08913 2/20 0.47
ADRA2B P18089 2/20 0.47
KCNH2 Q12809 1/20 0.47
HTR4 Q13639 1/20 0.47
MAP4K4 O95819 2/20 0.43
ACHE P22303 3/20 0.43
HRH3 Q9Y5N1 1/20 0.40
ADRA2C P18825 1/20 0.38
ATR Q13535 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12440015 0.88 MCHR1 (0.69) MCHR1ADRA2AADRA2BKCNH2HTR4
SCHEMBL2259794 0.82 ALDH1A1 (0.47) MCHR1ADRA2AADRA2BMAP4K4ADRA2C
SCHEMBL4804050 0.81 ALDH1A1 (0.50) MCHR1ADRA2AADRA2BACHEHRH3
Hydrochloric Acid SCHEMBL4809872 0.81 ALDH1A1 (0.46) MCHR1ADRA2AADRA2BMAP4K4ADRA2C
SCHEMBL1256258 0.79 ACHE (0.55) MCHR1MAP4K4ACHEHRH3
SCHEMBL18570582 0.76 APP (0.43) ADRA2AADRA2BADRA2C
SCHEMBL24618881 0.76 KIT (0.50) MCHR1ADRA2AADRA2BMAP4K4HRH3
SCHEMBL12441139 0.74 MCHR1 (0.55) MCHR1KCNH2ACHE
SCHEMBL3988708 0.73 BACE1 (0.50) MCHR1HRH3
SCHEMBL12440361 0.73 MCHR1 (0.54) MCHR1KCNH2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558578-B1 NOVEL ALKYNE COMPOUNDS HAVING AN MCH ANTAGONISTIC EFFECT AND MEDICAMENTS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM PHARMA (DE) 2013-03-13 EP disclosed