SCHEMBL14773

SCHEMBL14773

C=C(/C=C\C(=C/C)c1cc2cn(-c3ccc(CN4CC[C@@H](NC(=N)N)C4)cc3)c(=O)nc2[nH]1)S(=O)(=O)NC1CCNCC1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.33
CCR3 P51677 3/20 0.32
GRM2 Q14416 1/20 0.31
TEAD1 P28347 1/20 0.31
HTR1A P08908 1/20 0.31
CYP2D6 P10635 1/20 0.31
DRD2 P14416 1/20 0.31
HTR1D P28221 1/20 0.31
HTR2C P28335 1/20 0.31
HTR1F P30939 1/20 0.31
HTR2B P41595 1/20 0.31
HTR6 P50406 1/20 0.31
CYP3A43 Q9HB55 1/20 0.31
UTS2R Q9UKP6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20082562 0.79 ADORA2B (0.42) CCR3
SCHEMBL17277305 0.78 ROCK2 (0.40) ROCK2CCR3GRM2TEAD1DRD2
SCHEMBL12075449 0.76 CCR2 (0.39) ROCK2CCR3GRM2TEAD1DRD2
SCHEMBL12062170 0.76 ROCK2 (0.39) ROCK2CCR3GRM2TEAD1
SCHEMBL17277490 0.73 ROCK2 (0.46) ROCK2
SCHEMBL12075870 0.72 ROCK2 (0.45) ROCK2
SCHEMBL14775 0.72 TEAD1 (0.39) ROCK2CCR3GRM2TEAD1DRD2
SCHEMBL12062105 0.71 ADORA2B (0.35) ROCK2CCR3GRM2HTR1ACYP2D6
SCHEMBL12075462 0.71 ROCK2 (0.44) ROCK2
SCHEMBL12062108 0.68 ADORA2B (0.44) CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011047319-A2 ANTIMICROBIAL COMPOUNDS AND METHODS OF MAKING AND USING THE SAME RIB-X PHARMACEUTICALS, INC. (US) 2011-04-21 WO disclosed