SCHEMBL14775295

SCHEMBL14775295

CNCCC(c1ccc(OC)c(OC)c1)N1CCCCC1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
ACHE P22303 2/20 0.53
TSHR P16473 2/20 0.53
RAB9A P51151 1/20 0.53
SLC6A4 P31645 5/20 0.47
SLC6A2 P23975 4/20 0.47
SLC6A3 Q01959 4/20 0.47
P4HB P07237 1/20 0.44
POLB P06746 1/20 0.42
ATM Q13315 1/20 0.42
GAA P10253 1/20 0.41
TP53 P04637 1/20 0.40
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
TNF P01375 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14775491 0.87 ACHE (0.55) ALDH1A1ACHESLC6A4SLC6A2SLC6A3
SCHEMBL14775520 0.82 SLC6A2 (0.68) ALDH1A1ACHETSHRRAB9ASLC6A4
SCHEMBL14775125 0.74 SLC6A2 (0.51) ALDH1A1ACHETSHRRAB9ASLC6A4
SCHEMBL401565 0.73 SLC6A2 (0.67) ALDH1A1TSHRSLC6A4SLC6A2SLC6A3
Hydrochloric Acid SCHEMBL14775041 0.73 SLC6A2 (0.50) ALDH1A1ACHETSHRRAB9ASLC6A4
SCHEMBL19407169 0.73 PPARG (0.51) ALDH1A1ACHETSHRSLC6A4SLC6A2
SCHEMBL4786345 0.73 PPARG (0.51) ALDH1A1ACHETSHRSLC6A4SLC6A2
SCHEMBL14775127 0.69 SLC6A2 (0.66) ALDH1A1ACHESLC6A4SLC6A2SLC6A3
SCHEMBL9510573 0.69 ACHE (0.48) ALDH1A1ACHETSHRRAB9AMEN1
SCHEMBL9510568 0.69 ACHE (0.48) ALDH1A1ACHETSHRRAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2570409-B1 ARALKYL DIAMINE DERIVATIVES AND USES THEREOF AS ANTIDEPRESSANT SHANGHAI INST PHARM INDUSTRY (CN) 2015-07-08 EP claimed
US-8962621-B2 Aralkyl diamine derivatives and uses thereof as antidepressants SHANGHAI INSTITUTE OF PHARMACEUTICAL INDUSTRY (CN) 2015-02-24 US claimed
US-20130072488-A1 ARALKYL DIAMINE DERIVATIVES AND USES THEREOF AS ANTIDEPRESSANTS SHANGHAI INSTITUTE OF PHARMACEUTICAL INDUSTRY (CN) 2013-03-21 US claimed
EP-2570409-A1 ARALKYL DIAMINE DERIVATIVES AND USES THEREOF AS ANTIDEPRESSANT Shanghai Institute of Pharmaceutical Industry (CN) 2013-03-20 EP claimed
EP-2570409-B1 ARALKYL DIAMINE DERIVATIVES AND USES THEREOF AS ANTIDEPRESSANT SHANGHAI INST PHARM INDUSTRY (CN) 2015-07-08 EP disclosed
US-8962621-B2 Aralkyl diamine derivatives and uses thereof as antidepressants SHANGHAI INSTITUTE OF PHARMACEUTICAL INDUSTRY (CN) 2015-02-24 US disclosed
US-20130072488-A1 ARALKYL DIAMINE DERIVATIVES AND USES THEREOF AS ANTIDEPRESSANTS SHANGHAI INSTITUTE OF PHARMACEUTICAL INDUSTRY (CN) 2013-03-21 US disclosed
EP-2570409-A1 ARALKYL DIAMINE DERIVATIVES AND USES THEREOF AS ANTIDEPRESSANT Shanghai Institute of Pharmaceutical Industry (CN) 2013-03-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130072488-A1 ARALKYL DIAMINE DERIVATIVES AND USES THEREOF AS ANTIDEPRESSANTS MAOA, SLC6A2, MAOB ALDH1A1 390/4885ACHE 39/4885TSHR 2505/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.