SCHEMBL14775460

SCHEMBL14775460

COCCN1CCc2c[c]ccc2C1C(N)=O

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.36
PARP1 P09874 2/20 0.32
KDM4E B2RXH2 1/20 0.31
HDAC1 Q13547 1/20 0.30
HDAC8 Q9BY41 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2844323 0.89 HRH2 (0.32) KDM4EHDAC1HDAC8
SCHEMBL4748761 0.82 MAOA (0.32) OPRM1
SCHEMBL2844016 0.82 MTNR1A (0.38)
Hydrochloric Acid SCHEMBL4521946 0.81 MAOA (0.31) OPRM1KDM4E
SCHEMBL6969207 0.80 SIRT2 (0.39) OPRM1HDAC1HDAC8
SCHEMBL4514757 0.80 OPRK1 (0.32) OPRM1
Hydrochloric Acid SCHEMBL4504167 0.79 OPRK1 (0.32) OPRM1
SCHEMBL6961084 0.79 PRCP (0.39) KDM4E
SCHEMBL6960867 0.78 PARP1 (0.36) PARP1KDM4E
SCHEMBL6966047 0.78 ESR1 (0.37) PARP1HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951675-B1 TETRAHYDROISOQUINOLINE AS LXR MODULATORS BRISTOL MYERS SQUIBB CO (US) 2013-03-20 EP disclosed