SCHEMBL14775738

SCHEMBL14775738

O=C(Cc1ccc(C(F)(F)F)cc1)Nc1cc2ncccc2cc1O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.57
NLRP3 Q96P20 1/20 0.50
RIOK2 Q9BVS4 1/20 0.47
P2RX7 Q99572 2/20 0.46
ALDH1A1 P00352 1/20 0.45
CSNK1D P48730 2/20 0.44
P2RY14 Q15391 3/20 0.44
ANO1 Q5XXA6 2/20 0.44
MAPK8 P45983 1/20 0.43
MAPK10 P53779 1/20 0.43
EGLN1 Q9GZT9 1/20 0.43
TRPV1 Q8NER1 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
CLK1 P49759 1/20 0.43
GLS O94925 1/20 0.42
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2110907 0.79 EGLN1 (0.60) HDAC3NLRP3RIOK2P2RX7ALDH1A1
SCHEMBL15327088 0.76 KDM1A (0.53) P2RX7EGLN1
SCHEMBL14775742 0.74 P2RX7 (0.50) HDAC3P2RX7ALDH1A1KDM4EMAPT
SCHEMBL2108506 0.73 KDM4E (0.47) NLRP3RIOK2P2RX7ALDH1A1EGLN1
SCHEMBL29373364 0.72 MEN1 (0.61) NLRP3ALDH1A1CSNK1DKDM4EMAPT
SCHEMBL22246740 0.72 P2RX7 (0.47) NLRP3RIOK2P2RX7ALDH1A1CSNK1D
SCHEMBL13675951 0.71 MCHR1 (0.64) TRPV1
SCHEMBL29099861 0.71 MAPT (0.61) HDAC3RIOK2ALDH1A1CSNK1DP2RY14
SCHEMBL3958875 0.68 NPC1 (0.76) ALDH1A1EGLN1TRPV1MAPTMEN1
SCHEMBL28158289 0.68 MET (0.53) ALDH1A1KDM4EMAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963272-B1 HYDROXYQUINOLINE DERIVATIVES MERCK PATENT GMBH (DE) 2013-03-20 EP claimed
EP-1963272-B1 HYDROXYQUINOLINE DERIVATIVES MERCK PATENT GMBH (DE) 2013-03-20 EP disclosed