SCHEMBL148203

SCHEMBL148203

c1cncc(-c2cccc3c2[nH]c2ccccc23)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 5/20 0.65
CYP11B1 P15538 2/20 0.55
CYP11B2 P19099 1/20 0.55
PARP14 Q460N5 4/20 0.55
IDO1 P14902 2/20 0.50
LRRK2 Q5S007 1/20 0.50
HTR2B P41595 1/20 0.49
HTR5A P47898 1/20 0.49
KDM4E B2RXH2 3/20 0.49
ACHE P22303 1/20 0.49
GABRP O00591 1/20 0.49
GABRD O14764 1/20 0.49
IKBKB O14920 1/20 0.49
AURKA O14965 1/20 0.49
CHUK O15111 1/20 0.49
ALDH1A1 P00352 1/20 0.49
PIM1 P11309 1/20 0.49
TOP1 P11387 1/20 0.49
GABRA1 P14867 1/20 0.49
HPGD P15428 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29572015 1.00 TDO2 (0.65) TDO2CYP11B1CYP11B2PARP14IDO1
SCHEMBL28303023 0.94 TDO2 (0.62) TDO2CYP11B1CYP11B2PARP14IDO1
SCHEMBL28014781 0.91 TDO2 (0.59) TDO2CYP11B1CYP11B2PARP14IDO1
SCHEMBL29601793 0.84 TDO2 (0.49) TDO2PARP14IDO1HTR2BHTR5A
SCHEMBL28782760 0.84 TDO2 (0.49) TDO2PARP14IDO1HTR2BHTR5A
SCHEMBL28301583 0.84 TDO2 (0.60) TDO2CYP11B1CYP11B2PARP14IDO1
SCHEMBL26086391 0.83 TDO2 (0.49) TDO2PARP14IDO1HTR2BHTR5A
SCHEMBL28852044 0.82 IMPDH2 (0.53) TDO2PARP14IDO1HTR2BHTR5A
SCHEMBL191031 0.81 CDK4 (0.55) TDO2PARP14HTR2BHTR5AGABRP
SCHEMBL29412285 0.81 CDK4 (0.55) TDO2PARP14HTR2BHTR5AGABRP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109790117-A Carbazole benzene class fused-ring derivatives, polymer, mixture, composition, organic electronic device and preparation method thereof 广州华睿光电材料有限公司 2019-05-21 CN disclosed
US-8362065-B2 Carbazole carboxamide compounds useful as kinase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2013-01-29 US disclosed
US-20120058996-A1 CARBAZOLE CARBOXAMIDE COMPOUNDS USEFUL AS KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY 2012-03-08 US disclosed
US-8084620-B2 Carbazole carboxamide compounds useful as kinase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2011-12-27 US disclosed
US-20100160303-A1 CARBAZOLE CARBOXAMIDE COMPOUNDS USEFUL AS KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY 2010-06-24 US disclosed
CN-100348594-C Bidentate ligand and its iridium complex and electroluminescent device therewith UNIV WUHAN (CN) 2007-11-14 CN disclosed
CN-1680366-A Bidentate ligand and its iridium complex and electroluminescent device therewith UNIV WUHAN (CN) 2005-10-12 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120058996-A1 CARBAZOLE CARBOXAMIDE COMPOUNDS USEFUL AS KINASE INHIBITORS BTK, FLT3, JAK1 TDO2 2235/4885CYP11B1 2255/4885CYP11B2 2304/4885
US-20100160303-A1 CARBAZOLE CARBOXAMIDE COMPOUNDS USEFUL AS KINASE INHIBITORS BTK, FLT3, JAK1 TDO2 2235/4885CYP11B1 2255/4885CYP11B2 2304/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.