SCHEMBL1482214

SCHEMBL1482214

C=CC(CC(=O)Oc1ccccc1)N1CCC[Si]1(C)C

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.33
CYP2D6 P10635 3/20 0.33
CYP3A4 P08684 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
USP2 O75604 2/20 0.32
TSHR P16473 2/20 0.32
ALOX15 P16050 1/20 0.32
ALDH1A1 P00352 2/20 0.32
MGLL Q99685 1/20 0.32
CYP19A1 P11511 1/20 0.32
ELANE P08246 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
TEAD1 P28347 1/20 0.31
TEAD3 Q99594 1/20 0.31
MAPT P10636 1/20 0.31
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1478982 0.87
SCHEMBL1479020 0.83 CYP19A1 (0.35) GAACYP2D6TSHRALDH1A1MGLL
SCHEMBL1479075 0.71 ALDH1A1 (0.45) GAASMN1; SMN2TSHRALDH1A1MAPT
SCHEMBL1478900 0.69
SCHEMBL27678012 0.69 CYP19A1 (0.42) ALOX15ALDH1A1CYP19A1ELANEMAPT
SCHEMBL1479360 0.68 ALDH1A1 (0.37) GAASMN1; SMN2ALDH1A1MAPTMEN1
SCHEMBL8760983 0.68 CYP17A1 (0.35) CYP2D6CYP3A4TSHRALDH1A1CYP1A2
SCHEMBL3079292 0.65 ELANE (0.45) GAATSHRALDH1A1CYP19A1ELANE
SCHEMBL666155 0.65 POLB (0.47) GAACYP2D6TSHRALOX15ALDH1A1
SCHEMBL9113777 0.65 CYP19A1 (0.39) SMN1; SMN2ALDH1A1CYP19A1ELANEMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895670-B2 Functionalized polymers and methods for their manufacture BRIDGESTONE CORPORATION (JP) 2014-11-25 US claimed
US-20110077325-A1 FUNCTIONALIZED POLYMERS AND METHODS FOR THEIR MANUFACTURE BRIDGESTONE CORPORATION (JP) 2011-03-31 US claimed
EP-2699606-B1 POLYMERS FUNCTIONALIZED WITH A CARBOXYLIC OR THIOCARBOXYLIC ESTER CONTAINING A SILYLATED AMINO GROUP BRIDGESTONE CORP (JP) 2016-09-28 EP disclosed
US-9403919-B2 Polymers functionalized with a carboxylic or thiocarboxylic ester containing a silylated amino group BRIDGESTONE CORPORATION (JP) 2016-08-02 US disclosed
US-8895670-B2 Functionalized polymers and methods for their manufacture BRIDGESTONE CORPORATION (JP) 2014-11-25 US disclosed
EP-2483317-B1 FUNCTIONALIZED POLYMERS AND METHODS FOR THEIR MANUFACTURE BRIDGESTONE CORP (JP) 2014-02-26 EP disclosed
EP-2699606-A2 POLYMERS FUNCTIONALIZED WITH A CARBOXYLIC OR THIOCARBOXYLIC ESTER CONTAINING A SILYLATED AMINO GROUP Bridgestone Corporation (JP) 2014-02-26 EP disclosed
US-20140018500-A1 Polymers Functionalized With A Carboxylic Or Thiocarboxylic Ester Containing A Silylated Amino Group BRIDGESTONE CORPORATION (JP) 2014-01-16 US disclosed
WO-2012135451-A2 POLYMERS FUNCTIONALIZED WITH A CARBOXYLIC OR THIOCARBOXYLIC ESTER CONTAINING A SILYLATED AMINO GROUP BRIDGESTONE CORPORATION (JP) 2012-10-04 WO disclosed
EP-2483317-A1 FUNCTIONALIZED POLYMERS AND METHODS FOR THEIR MANUFACTURE Bridgestone Corporation (JP) 2012-08-08 EP disclosed
US-20120184677-A1 FUNCTIONALIZED POLYMERS AND METHODS FOR THEIR MANUFACTURE BRIDGESTONE CORPORATION (JP) 2012-07-19 US disclosed
WO-2011041534-A1 FUNCTIONALIZED POLYMERS AND METHODS FOR THEIR MANUFACTURE BRIDGESTONE CORPORATION (JP) 2011-04-07 WO disclosed
US-20110077325-A1 FUNCTIONALIZED POLYMERS AND METHODS FOR THEIR MANUFACTURE BRIDGESTONE CORPORATION (JP) 2011-03-31 US disclosed