SCHEMBL8760983

SCHEMBL8760983

C=CC(c1ccccc1)N1CCC[Si]1(C)C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.35
CYP2D6 P10635 8/20 0.33
KCNH2 Q12809 6/20 0.33
CYP1A2 P05177 5/20 0.33
CYP3A4 P08684 5/20 0.33
CYP2C19 P33261 5/20 0.33
CYP2C9 P11712 4/20 0.33
KCNA5 P22460 4/20 0.33
KCNE1 P15382 1/20 0.33
OPRD1 P41143 1/20 0.32
ALDH1A1 P00352 1/20 0.31
MCOLN3 Q8TDD5 1/20 0.31
TSHR P16473 1/20 0.31
CHRM2 P08172 2/20 0.31
ADRA2A P08913 2/20 0.31
CHRM1 P11229 2/20 0.31
DRD1 P21728 2/20 0.31
OPRM1 P35372 2/20 0.31
DRD3 P35462 2/20 0.31
SLC6A3 Q01959 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774648 0.72 OPRD1 (0.37) CYP17A1CYP2D6KCNH2OPRD1CHRM2
SCHEMBL3294321 0.71 CYP2D6 (0.55) CYP17A1CYP2D6KCNH2CYP1A2CYP3A4
SCHEMBL2579537 0.70 CYP2D6 (0.48) CYP17A1CYP2D6KCNH2CYP1A2CYP3A4
SCHEMBL11136769 0.69 CYP1A2 (0.57) CYP2D6KCNH2CYP1A2CYP3A4CYP2C19
SCHEMBL6837651 0.69 CYP1A2 (0.57) CYP2D6KCNH2CYP1A2CYP3A4CYP2C19
SCHEMBL6838012 0.69 CYP1A2 (0.57) CYP2D6KCNH2CYP1A2CYP3A4CYP2C19
SCHEMBL30518149 0.69 CYP1A2 (0.57) CYP2D6KCNH2CYP1A2CYP3A4CYP2C19
SCHEMBL6837652 0.69 CYP1A2 (0.57) CYP2D6KCNH2CYP1A2CYP3A4CYP2C19
SCHEMBL2361182 0.69 CYP1A2 (0.57) CYP2D6KCNH2CYP1A2CYP3A4CYP2C19
SCHEMBL986928 0.67 CYP2D6 (0.59) CYP2D6KCNH2CYP3A4CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0578186-B1 Method for the preparation of 1-aza-2-silacyclopentane compounds DOW CORNING KK (JP) 1997-06-04 EP disclosed
US-5281736-A Method for the preparation of 1-aza-2-silacyclopentane compounds DOW CORNING JAPAN, LTD. (JP) 1994-01-25 US disclosed
EP-0578186-A1 Method for the preparation of 1-AZA-2-silacyclopentane compounds DOW CORNING JAPAN, LTD. (JP) 1994-01-12 EP disclosed