SCHEMBL14823736

SCHEMBL14823736

CC(=O)c1ccc(C)c(-c2ccc(C#N)cc2)c1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 6/20 0.56
ALDH1A1 P00352 1/20 0.49
MAPT P10636 1/20 0.49
HSD17B1 P14061 1/20 0.46
KDM1A O60341 7/20 0.44
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
SLC22A12 Q96S37 1/20 0.43
MAP4K4 O95819 1/20 0.43
NSD2 O96028 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1231896 0.88 SLC22A12 (0.56) MAPK14KDM1ACA1CA2SLC22A12
SCHEMBL2428847 0.84 MAPK14 (0.52) MAPK14ALDH1A1KDM1AMAP4K4
SCHEMBL2039607 0.81 SLC22A12 (0.53) MAPK14SLC22A12MAP4K4
SCHEMBL17855536 0.80 MAPT (0.48) ALDH1A1MAPTHSD17B1KDM1ACA1
SCHEMBL10058042 0.79 MAPT (0.66) ALDH1A1MAPTHSD17B1CA1CA2
SCHEMBL163209 0.77 ALDH1A1 (0.72) ALDH1A1MAPTCA1CA2
SCHEMBL1140572 0.76 MAPK14 (0.64) MAPK14
SCHEMBL10110951 0.76 ALDH1A1 (0.56) MAPK14ALDH1A1KDM1A
SCHEMBL27885275 0.76 HSD17B1 (0.44) MAPK14MAPTHSD17B1
SCHEMBL2345404 0.76 HRH2 (0.47) MAPK14ALDH1A1MAPTCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2021328-B1 COMPOUNDS AND COMPOSITIONS AS HEDGEHOG PATHWAY MODULATORS IRM LLC (BM) 2013-04-03 EP disclosed