SCHEMBL17855536

SCHEMBL17855536

CC(=O)c1ccc(-c2ccc(C#N)cc2)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.48
ALDH1A1 P00352 2/20 0.48
KDM1A O60341 4/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
GAA P10253 1/20 0.45
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
P4HB P07237 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
SLC6A9 P48067 1/20 0.42
SLC6A5 Q9Y345 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
SLC22A12 Q96S37 1/20 0.42
MAP4K4 O95819 1/20 0.42
RARB P10826 1/20 0.42
HSD17B1 P14061 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19656582 0.84 GSK3B (0.45) MAPTALDH1A1KDM1ASMN1; SMN2GAA
SCHEMBL14823736 0.80 MAPK14 (0.56) MAPTALDH1A1KDM1ACA1CA2
SCHEMBL15999132 0.80 MAP4K4 (0.52) PDE3BPDE3ASLC22A12MAP4K4RARB
SCHEMBL10269902 0.79 PTGS1 (0.55) MAPTSMN1; SMN2SLC6A9RARBNPC1
SCHEMBL15605814 0.78 GAPDH (0.44) MAPTALDH1A1KDM1ASMN1; SMN2GAA
SCHEMBL16844139 0.78 PDE3B (0.42) KDM1APDE3BPDE3ASLC22A12
SCHEMBL10058042 0.78 MAPT (0.66) MAPTALDH1A1SMN1; SMN2CA1CA2
SCHEMBL2559215 0.78 RARB (0.59) MAPTALDH1A1SMN1; SMN2CA1CA2
SCHEMBL5142555 0.77 CYP2C19 (0.58) SMN1; SMN2CA1CA2MAP4K4NPC1
SCHEMBL397141 0.77 KIF11 (0.61) PDE3BPDE3ACYP11B1CYP11B2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016096081-A1 BIMESOGENIC COMPOUNDS AND MESOGENIC MEDIA MERCK PATENT GMBH (DE) 2016-06-23 WO disclosed