SCHEMBL14844388

SCHEMBL14844388

NN(C(=O)C1CCCCC1)c1ccon1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.37
LMNA P02545 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
HPGD P15428 2/20 0.34
PTPN1 P18031 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
OPRD1 P41143 1/20 0.34
NPC1 O15118 4/20 0.33
RAB9A P51151 4/20 0.33
ALDH1A1 P00352 2/20 0.33
USP2 O75604 1/20 0.33
HSD17B10 Q99714 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14844279 0.73 SMN1; SMN2 (0.36) LMNASMN1; SMN2HPGDPTPN1HDAC3
SCHEMBL22496063 0.71 ALDH1A1 (0.40) LMNASMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL2464249 0.69 HTT (0.50) LMNASMN1; SMN2HPGDHDAC3HDAC1
Hydrochloric Acid SCHEMBL11830306 0.68 HTT (0.49) LMNASMN1; SMN2HPGDHDAC3HDAC1
SCHEMBL20268246 0.67 HTT (0.51) LMNASMN1; SMN2HPGDHDAC3HDAC1
SCHEMBL6425135 0.67 CNR2 (0.52) SMN1; SMN2HPGDNPSR1NPC1RAB9A
SCHEMBL2592597 0.66 ALDH1A1 (0.44) SMN1; SMN2HDAC3HDAC1HDAC2NPSR1
SCHEMBL19265536 0.65 CNR2 (0.50) SMN1; SMN2HPGDNPC1RAB9AALDH1A1
SCHEMBL2259800 0.64 HTT (0.51) LMNASMN1; SMN2HPGDNPSR1NPC1
SCHEMBL11569306 0.61 TRPM8 (0.36) NPC1RAB9AALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2763997-A1 CYCLOHEXYL-4H,6H-5-OXA-2,3,10B-TRIAZA-BENZO[E]AZULENES AS V1A ANTAGONISTS F.HOFFMANN-LA ROCHE AG (CH) 2014-08-13 EP disclosed
WO-2013050334-A1 CYCLOHEXYL-4H,6H-5-OXA-2,3,10B-TRIAZA-BENZO[E]AZULENES AS V1A ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2013-04-11 WO disclosed