SCHEMBL14850872

SCHEMBL14850872

COc1ccccc1-c1ccc(C)cc1C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.55
AKR1C2 P52895 1/20 0.55
S1PR1 P21453 2/20 0.48
HTR7 P34969 4/20 0.47
ACHE P22303 1/20 0.47
APP P05067 1/20 0.46
PTPRC P08575 1/20 0.45
PTPN1 P18031 1/20 0.45
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA4 P22748 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
HPGD P15428 3/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5184745 0.88 ACHE (0.56) AKR1C3AKR1C2HTR7ACHEAPP
SCHEMBL16542335 0.86 ACHE (0.58) AKR1C3AKR1C2ACHEHPGDCYP3A4
SCHEMBL13069497 0.85 ACHE (0.52) AKR1C3AKR1C2S1PR1HTR7ACHE
SCHEMBL277907 0.85 HTR7 (0.59) AKR1C3AKR1C2HTR7ACHEAPP
SCHEMBL4231404 0.81 AKR1C3 (0.52) AKR1C3AKR1C2S1PR1HTR7APP
SCHEMBL27537379 0.81 AKR1C3 (0.52) AKR1C3AKR1C2S1PR1HTR7APP
SCHEMBL27533596 0.81 AKR1C3 (0.52) AKR1C3AKR1C2S1PR1HTR7APP
SCHEMBL27555994 0.81 AKR1C3 (0.52) AKR1C3AKR1C2S1PR1HTR7APP
SCHEMBL321430 0.81 CA1 (0.55) AKR1C3AKR1C2S1PR1HTR7APP
SCHEMBL3958057 0.81 ACHE (0.52) S1PR1HTR7ACHEHPGDCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013050938-A1 3,7-DIAZABICYCLO[3.3.1]NONANE AND 9-OXA-3,7-DIAZABICYCLO[3.3.1]NONANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2013-04-11 WO disclosed