SCHEMBL14856552

SCHEMBL14856552

CCCCOC(=O)O[C@@]1(NC(=O)c2cncc(N)c2)CCOC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.33
SLC6A5 Q9Y345 2/20 0.33
LMNA P02545 4/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TSHR P16473 1/20 0.33
PDE4D Q08499 1/20 0.33
P2RX3 P56373 1/20 0.33
SPHK1 Q9NYA1 4/20 0.32
ALDH1A1 P00352 3/20 0.32
MAPT P10636 3/20 0.32
BDKRB1 P46663 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
DDO Q99489 1/20 0.32
DGAT2 Q96PD7 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10070601 0.83 SPHK1 (0.37) HTR2ASLC6A5LMNACYP1A2CYP3A4
SCHEMBL185855 0.82 KDM4E (0.41) LMNAALDH1A1BDKRB1KDM4EMEN1
SCHEMBL200210 0.80 HTR2A (0.33) HTR2ASLC6A5LMNACYP1A2CYP3A4
SCHEMBL186114 0.73 KDM4E (0.43) LMNACYP1A2ALDH1A1BDKRB1KDM4E
SCHEMBL11984274 0.72 BDKRB1 (0.39) LMNAALDH1A1BDKRB1KDM4EMEN1
SCHEMBL185854 0.70 KDM4E (0.45) LMNAL3MBTL1TSHRALDH1A1BDKRB1
SCHEMBL2805627 0.70 KDM4E (0.45) LMNAL3MBTL1TSHRALDH1A1BDKRB1
SCHEMBL14856657 0.70 KDM4E (0.45) L3MBTL1ALDH1A1KDM4EDGAT2SMN1; SMN2
SCHEMBL185596 0.67 VNN1 (0.38) BDKRB1DGAT2
SCHEMBL2787463 0.67 VNN1 (0.38) BDKRB1DGAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed