SCHEMBL14865000

SCHEMBL14865000

COc1ccc(-c2ccc(CCC(=O)O)n2NC(N)=O)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 13/20 1.00
ALDH1A1 P00352 12/20 0.72
HSD17B10 Q99714 5/20 0.72
POLB P06746 4/20 0.72
PKM P14618 2/20 0.72
TSHR P16473 1/20 0.72
RECQL P46063 1/20 0.72
MEN1 O00255 4/20 0.68
KMT2A Q03164 4/20 0.68
LMNA P02545 2/20 0.68
TDP1 Q9NUW8 2/20 0.68
MAPT P10636 10/20 0.67
GAA P10253 4/20 0.63
HPGD P15428 3/20 0.63
ALOX15 P16050 3/20 0.63
CASP1 P29466 2/20 0.63
USP2 O75604 1/20 0.63
ALOX12 P18054 1/20 0.63
CASP7 P55210 1/20 0.63
NPSR1 Q6W5P4 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20248226 0.85 KDM4E (0.79) KDM4EALDH1A1HSD17B10POLBPKM
SCHEMBL20250909 0.84 KDM4E (1.00) KDM4EALDH1A1HSD17B10POLBPKM
SCHEMBL14865018 0.80 KDM4E (0.85) KDM4EALDH1A1HSD17B10POLBPKM
SCHEMBL19275255 0.80 ALDH1A1 (0.77) KDM4EALDH1A1HSD17B10POLBPKM
SCHEMBL14865002 0.76 KDM4E (0.86) KDM4EALDH1A1HSD17B10POLBPKM
SCHEMBL20248183 0.75 KDM4E (0.79) KDM4EALDH1A1HSD17B10POLBPKM
SCHEMBL242401 0.74 PTGS1 (0.62) KDM4EALDH1A1HSD17B10POLBPKM
SCHEMBL243617 0.74 MAPT (0.74) KDM4EALDH1A1HSD17B10POLBMEN1
SCHEMBL14865007 0.73 MAPT (1.00) KDM4EALDH1A1HSD17B10POLBMEN1
SCHEMBL15862515 0.73 MAPT (0.72) KDM4EALDH1A1HSD17B10POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2581451-A1 Compounds for inhibiting mammalian s-nitrosoglutathione reductase Indiana University Research and Technology Corporation (US) 2013-04-17 EP disclosed