SCHEMBL14865109

SCHEMBL14865109

C[C@@H](c1ccc(Br)cc1)N(CCCc1ccc(F)cc1)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
SLC6A4 P31645 2/20 0.40
SLC6A3 Q01959 2/20 0.40
SLC6A2 P23975 1/20 0.40
ALOX5 P09917 1/20 0.40
AGTR2 P50052 3/20 0.39
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
TRPM8 Q7Z2W7 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13077090 0.87 SLC6A4 (0.42) SLC6A4SLC6A3SLC6A2ALOX5
SCHEMBL12767085 0.86 SLC6A2 (0.40) KMT2ASLC6A4SLC6A3SLC6A2AGTR2
SCHEMBL12767088 0.84 ALOX5 (0.40) SLC6A4SLC6A3SLC6A2ALOX5AGTR2
SCHEMBL3637292 0.83 NPC1 (0.47) MEN1KMT2ASLC6A4SLC6A3SLC6A2
SCHEMBL3408775 0.82 ALOX5 (0.41) MEN1KMT2AALOX5TRPM8TDP1
SCHEMBL3408769 0.82 ALOX5 (0.41) MEN1KMT2AALOX5TRPM8TDP1
SCHEMBL3408772 0.82 ALOX5 (0.41) MEN1KMT2AALOX5TRPM8TDP1
SCHEMBL18380905 0.81 ALDH1A1 (0.39) SLC6A4SLC6A3SLC6A2
SCHEMBL13953697 0.80 ALOX5 (0.37) ALOX5TRPM8
SCHEMBL16791621 0.79 ALOX5 (0.39) ALOX5TRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2300461-B1 CYCLIC INHIBITORS OF 11BETA-HYDROXYSTEROID DEHYDROGENASE 1 VITAE PHARMACEUTICALS INC (US) 2013-04-17 EP disclosed