SCHEMBL14865312

SCHEMBL14865312

C=C(NCc1ccc(Nc2ccccc2C(F)(F)F)cc1)C1(NC(=O)C2CC2)CC1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.41
EPHX2 P34913 4/20 0.38
MAPT P10636 2/20 0.38
CYP2C9 P11712 2/20 0.36
SCN9A Q15858 1/20 0.36
SSTR4 P31391 1/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
KMT2A Q03164 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2806172 0.91 POLB (0.43) POLBEPHX2MAPTCYP2C9SCN9A
SCHEMBL13128411 0.83 POLB (0.45) POLBEPHX2MAPTCYP2C9MEN1
SCHEMBL13128471 0.81 CTDSP1 (0.39) POLBEPHX2MAPTCYP2C9SCN9A
SCHEMBL2809250 0.78 ALDH1A1 (0.41) POLBMAPTCYP2C9ALDH1A1HPGD
SCHEMBL185966 0.78 BDKRB1 (0.40) POLBMAPTCYP2C9ALDH1A1HPGD
SCHEMBL2806680 0.78 RAB9A (0.39) POLBCYP2C9MEN1KMT2AGAA
SCHEMBL13128461 0.78 CTDSP1 (0.36) POLBEPHX2CYP2C9SCN9A
SCHEMBL185673 0.77 POLB (0.45) POLBEPHX2MAPTCYP2C9USP2
SCHEMBL2806861 0.77 SMN1; SMN2 (0.40) POLBEPHX2SCN9ASSTR4MEN1
SCHEMBL2807722 0.76 CTSL (0.44) POLBEPHX2MAPTALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed