SCHEMBL14865327

SCHEMBL14865327

CC1(C(=O)NCc2ccc(Nc3ccc(Cl)cc3C(F)(F)F)cn2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HTT P42858 1/20 0.39
PAX8 Q06710 1/20 0.39
P2RX7 Q99572 1/20 0.39
CNR2 P34972 6/20 0.39
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TRPV1 Q8NER1 2/20 0.38
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
BACE1 P56817 1/20 0.37
PTGES O14684 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14865300 0.90 TRPA1 (0.41) P2RX7CNR2BACE1PTGES
SCHEMBL2805697 0.89 RAB9A (0.41) RAB9ACYP1A2CYP2D6CYP2C19KDM4E
SCHEMBL2780230 0.87 CNR2 (0.40) RAB9ACYP1A2CYP2D6CYP2C19KDM4E
SCHEMBL2809946 0.86 CNR2 (0.39) RAB9ACYP1A2CYP2D6CYP2C19KDM4E
Trifluoroacetic Acid SCHEMBL2809036 0.86 RAB9A (0.38) RAB9ACYP1A2CYP2D6CYP2C19KDM4E
SCHEMBL2807298 0.85 CNR2 (0.40) RAB9ACYP1A2CYP2D6CYP2C19KDM4E
SCHEMBL19418576 0.85 CNR2 (0.39) RAB9ACYP1A2CYP2D6CYP2C19KDM4E
SCHEMBL13159819 0.84 CNR2 (0.38) RAB9ACYP1A2CYP2D6CYP2C19KDM4E
SCHEMBL2811071 0.84 RAB9A (0.44) RAB9ACYP1A2CYP2D6CYP2C19KDM4E
SCHEMBL2809043 0.84 CNR2 (0.38) RAB9ACYP1A2CYP2D6CYP2C19KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed