SCHEMBL14865300

SCHEMBL14865300

CC1(C(=O)NCc2ccc(Nc3ccc(F)cc3C(F)(F)F)cn2)CC1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 8/20 0.41
P2RX7 Q99572 2/20 0.39
CNR2 P34972 1/20 0.38
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
BACE1 P56817 1/20 0.36
NTRK1 P04629 1/20 0.35
AURKA O14965 2/20 0.35
OPRL1 P41146 1/20 0.35
PTGES O14684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14865327 0.90 RAB9A (0.40) P2RX7CNR2BACE1PTGES
SCHEMBL2807472 0.89 P2RX7 (0.39) TRPA1P2RX7CNR2HDAC3HDAC1
Hydrochloric Acid SCHEMBL2805225 0.88 P2RX7 (0.39) TRPA1P2RX7CNR2HDAC3HDAC1
SCHEMBL2782482 0.86 P2RX7 (0.38) TRPA1P2RX7CNR2HDAC3HDAC1
SCHEMBL2812751 0.85 P2RX7 (0.37) TRPA1P2RX7CNR2HDAC3HDAC1
SCHEMBL19418572 0.85 CNR2 (0.38) TRPA1P2RX7CNR2HDAC3HDAC1
SCHEMBL19418558 0.85 TRPA1 (0.37) TRPA1P2RX7CNR2HDAC3HDAC1
SCHEMBL2805100 0.83 CNR2 (0.37) TRPA1P2RX7CNR2AURKAOPRL1
SCHEMBL2809823 0.83 CNR2 (0.37) TRPA1P2RX7CNR2AURKAOPRL1
SCHEMBL13160253 0.83 TRPA1 (0.36) TRPA1P2RX7CNR2BACE1NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed