SCHEMBL14865331

SCHEMBL14865331

O=C(N[C@@]1(C(=O)NCc2ncc(Nc3ccccc3C(F)(F)F)cc2Cl)CCOC1)c1cn[nH]c1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.34
ROCK1 Q13464 2/20 0.34
NAMPT P43490 2/20 0.33
BDKRB1 P46663 1/20 0.33
P2RX7 Q99572 4/20 0.33
CNR1 P21554 1/20 0.32
MAPK1 P28482 1/20 0.32
CTDSP1 Q9GZU7 1/20 0.32
CNR2 P34972 2/20 0.32
ACACB O00763 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPK9 P45984 1/20 0.31
MAPK10 P53779 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2805217 0.89 P2RX7 (0.36) BDKRB1P2RX7CTDSP1CNR2HTT
SCHEMBL197308 0.87 BDKRB1 (0.36) BDKRB1P2RX7CTDSP1CNR2HTT
SCHEMBL2808176 0.87 BDKRB1 (0.36) BDKRB1P2RX7CTDSP1CNR2HTT
SCHEMBL10066086 0.83 CNR2 (0.36) P2RX7CNR1CNR2KDM4E
SCHEMBL15460097 0.83 ALOX15 (0.36) P2RX7CNR1MAPK1CNR2
SCHEMBL186187 0.83 TRPV1 (0.36) P2RX7CTDSP1HTT
SCHEMBL2805848 0.82 BDKRB1 (0.39) BDKRB1CNR2
SCHEMBL10071820 0.82 EPHX2 (0.33) ROCK2ROCK1BDKRB1P2RX7CNR2
SCHEMBL2805120 0.82 CNR2 (0.38) BDKRB1P2RX7CNR1CNR2KDM4E
SCHEMBL2809983 0.82 OPRL1 (0.36) BDKRB1CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed