SCHEMBL14865400

SCHEMBL14865400

Cc1ncc(C(=O)N[C@@]2(C(=O)NCc3ccc(Nc4ccccc4C(C)(F)F)cc3F)CCOC2)cn1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 8/20 0.34
CNR1 P21554 1/20 0.34
EPHX2 P34913 1/20 0.32
PDE2A O00408 1/20 0.32
NTRK1 P04629 1/20 0.32
HDAC6 Q9UBN7 1/20 0.31
MAPK9 P45984 2/20 0.31
MAPK10 P53779 2/20 0.31
P2RX7 Q99572 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
CXCR2 P25025 1/20 0.31
RAF1 P04049 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2811762 0.95 BDKRB1 (0.35) BDKRB1CNR1EPHX2PDE2ANTRK1
SCHEMBL2806388 0.88 HDAC3 (0.38) BDKRB1EPHX2NTRK1HDAC6P2RX7
SCHEMBL2811531 0.88 BDKRB1 (0.37) BDKRB1CNR1NTRK1P2RX7RAF1
SCHEMBL2805174 0.87 BDKRB1 (0.41) BDKRB1CNR1NTRK1HDAC6MAPK9
SCHEMBL10070758 0.86 EPHX2 (0.40) BDKRB1EPHX2P2RX7
SCHEMBL185850 0.84 FAAH (0.38) BDKRB1CNR1EPHX2NTRK1MAPK9
SCHEMBL2809623 0.84 BDKRB1 (0.39) BDKRB1HDAC6MAPK9MAPK10
SCHEMBL185861 0.82 BDKRB1 (0.37) BDKRB1CNR1EPHX2
SCHEMBL16404411 0.81 ROCK2 (0.34) BDKRB1CXCR2
SCHEMBL9892777 0.81 PTGES (0.34) BDKRB1CNR1EPHX2MAPK9MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed