SCHEMBL14865402

SCHEMBL14865402

N#Cc1ccc(C(=O)NC2(C(=O)NCc3ccc(Nc4ccc(F)cc4C(F)(F)S)cn3)CC2)cn1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 1/20 0.36
KCNQ2 O43526 1/20 0.36
AR P10275 6/20 0.35
CTSK P43235 4/20 0.34
CTSS P25774 3/20 0.34
EPHX2 P34913 1/20 0.34
RORC P51449 1/20 0.33
SCN10A Q9Y5Y9 1/20 0.33
CTSL P07711 1/20 0.33
PRKAA2 P54646 2/20 0.32
CHEK1 O14757 2/20 0.32
TRPA1 O75762 1/20 0.31
BDKRB1 P46663 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL186506 0.94 AR (0.38) KCNQ3KCNQ2ARCTSKCTSS
SCHEMBL186730 0.83 TRPA1 (0.40) TRPA1BDKRB1
SCHEMBL186050 0.82 CNR1 (0.36) KCNQ3KCNQ2TRPA1BDKRB1
SCHEMBL186398 0.82 HDAC1 (0.35) ARCTSKCTSSEPHX2CTSL
SCHEMBL186387 0.82 KCNQ3 (0.42) KCNQ3KCNQ2BDKRB1
SCHEMBL185570 0.82 ALDH1A1 (0.36) TRPA1BDKRB1
SCHEMBL2807486 0.81 HDAC3 (0.41) TRPA1BDKRB1
SCHEMBL2811921 0.80 HDAC3 (0.38) CTSKCTSSTRPA1BDKRB1
SCHEMBL185915 0.80 ABL1 (0.38) CTSKCTSSBDKRB1
SCHEMBL2805859 0.80 BDKRB1 (0.41) ARTRPA1BDKRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed