SCHEMBL14865417

SCHEMBL14865417

CN(c1ccc(CNC(=O)[C@]2(NC(=O)c3cn[nH]c(=O)c3)CCOC2)c(F)c1)c1ccccc1C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.34
BDKRB1 P46663 4/20 0.33
CNR1 P21554 1/20 0.32
TRPV1 Q8NER1 1/20 0.31
AR P10275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9892777 0.85 PTGES (0.34) BDKRB1CNR1TRPV1
SCHEMBL2805106 0.80 AURKA (0.35) HDAC6CNR1
SCHEMBL2806442 0.79 P2RX7 (0.33) CNR1
SCHEMBL10070731 0.79 EPHX2 (0.38)
SCHEMBL2807318 0.78 BDKRB1 (0.39) BDKRB1TRPV1
SCHEMBL19418557 0.77 OPRL1 (0.33)
SCHEMBL2808594 0.74 OPRL1 (0.36) BDKRB1
SCHEMBL14856801 0.73 TRPV1 (0.34) BDKRB1CNR1TRPV1
SCHEMBL15460053 0.73 OPRL1 (0.34) HDAC6
SCHEMBL16404399 0.73 ROCK2 (0.33) BDKRB1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed