SCHEMBL14865486

SCHEMBL14865486

N/C=C(\S)C(=O)N[C@@]1(C(=O)NCc2ccc(Nc3ccc(F)cc3C(F)(F)F)cc2)CCOC1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 5/20 0.38
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
CNR2 P34972 5/20 0.33
CNR1 P21554 2/20 0.33
HDAC1 Q13547 1/20 0.32
TRPV1 Q8NER1 1/20 0.31
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA7 P43166 1/20 0.30
CA9 Q16790 1/20 0.30
P2RX7 Q99572 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14865447 0.92 ALDH1A1 (0.36) OPRL1ALDH1A1LMNACNR2CNR1
SCHEMBL14865314 0.86 CNR2 (0.34) OPRL1CNR2CNR1HDAC1CA1
SCHEMBL2813417 0.82 BDKRB1 (0.41) OPRL1ALDH1A1LMNACNR2HDAC1
SCHEMBL13128639 0.81 BDKRB1 (0.40) OPRL1ALDH1A1LMNACNR2HDAC1
SCHEMBL186503 0.81 CNR2 (0.37) OPRL1ALDH1A1CNR2HDAC1
SCHEMBL2811657 0.81 CNR2 (0.37) OPRL1ALDH1A1CNR2HDAC1
SCHEMBL2809544 0.81 OPRL1 (0.39) OPRL1ALDH1A1CNR2HDAC1
SCHEMBL2805738 0.81 AR (0.39) OPRL1ALDH1A1LMNACNR2CNR1
SCHEMBL2804935 0.80 OPRL1 (0.38) OPRL1CNR2CNR1HDAC1CA1
SCHEMBL2808552 0.80 PTK2 (0.41) OPRL1CNR2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed