SCHEMBL14865447

SCHEMBL14865447

N/C=C(\S)C(=O)NC1(C(=O)NCc2ccc(Nc3ccc(F)cc3C(F)(F)F)cc2)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
CNR2 P34972 3/20 0.35
CNR1 P21554 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
BDKRB1 P46663 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
P2RX7 Q99572 2/20 0.33
OPRL1 P41146 2/20 0.33
MTOR P42345 1/20 0.32
HDAC1 Q13547 1/20 0.32
OPRM1 P35372 1/20 0.32
AURKA O14965 2/20 0.32
POLB P06746 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14865314 0.92 CNR2 (0.34) CNR2CNR1CA1CA2CA7
SCHEMBL14865486 0.92 OPRL1 (0.38) ALDH1A1LMNACNR2CNR1CA1
SCHEMBL184742 0.85 CYP3A4 (0.40) ALDH1A1LMNACNR2CNR1CYP3A4
SCHEMBL185221 0.82 ALDH1A1 (0.38) ALDH1A1LMNACNR2CNR1CYP3A4
SCHEMBL14865381 0.81 CNR2 (0.35) ALDH1A1CNR2CYP2C19P2RX7RAB9A
SCHEMBL2808499 0.80 ALDH1A1 (0.40) ALDH1A1LMNACNR2CYP3A4CYP2C9
SCHEMBL13128425 0.80 BDKRB1 (0.48) ALDH1A1LMNACNR2CNR1CYP3A4
SCHEMBL2807564 0.80 LMNA (0.37) ALDH1A1LMNACNR2CNR1CYP3A4
SCHEMBL185133 0.80 CNR2 (0.41) ALDH1A1CNR2CNR1CA1CA2
SCHEMBL186467 0.79 AR (0.41) ALDH1A1LMNACNR2CNR1BDKRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed