SCHEMBL14865314

SCHEMBL14865314

C=C(NCc1ccc(Nc2ccc(F)cc2C(F)(F)F)cc1)C1(NC(=O)/C(S)=C/N)CC1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 3/20 0.34
CNR1 P21554 2/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
HDAC1 Q13547 1/20 0.31
BTK Q06187 1/20 0.31
MTOR P42345 1/20 0.31
PTK2 Q05397 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRL1 P41146 1/20 0.31
AURKA O14965 2/20 0.30
NAMPT P43490 1/20 0.30
POLB P06746 1/20 0.30
RAB9A P51151 1/20 0.30
P2RX7 Q99572 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14865447 0.92 ALDH1A1 (0.36) CNR2CNR1CA1CA2CA7
SCHEMBL14865486 0.86 OPRL1 (0.38) CNR2CNR1CA1CA2CA7
SCHEMBL184742 0.77 CYP3A4 (0.40) CNR2CNR1CA1CA2CA7
SCHEMBL185133 0.76 CNR2 (0.41) CNR2CNR1CA1CA2CA7
SCHEMBL185221 0.75 ALDH1A1 (0.38) CNR2CNR1CA1CA2CA7
SCHEMBL14865381 0.74 CNR2 (0.35) CNR2RAB9AP2RX7
SCHEMBL2808499 0.73 ALDH1A1 (0.40) CNR2OPRL1AURKAP2RX7
SCHEMBL13128425 0.73 BDKRB1 (0.48) CNR2CNR1HDAC1PTK2AURKA
SCHEMBL2807564 0.73 LMNA (0.37) CNR2CNR1OPRL1NAMPTPOLB
SCHEMBL186467 0.72 AR (0.41) CNR2CNR1HDAC1PTK2AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed