SCHEMBL14879772

SCHEMBL14879772

COC(=O)c1cc(N)c(Oc2ccccc2)c(C(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.45
NOTUM Q6P988 2/20 0.44
ALDH1A1 P00352 4/20 0.42
KDM4E B2RXH2 3/20 0.42
GAA P10253 3/20 0.42
HPGD P15428 3/20 0.42
PKM P14618 1/20 0.42
CFTR P13569 5/20 0.42
TSHR P16473 1/20 0.41
MAPT P10636 2/20 0.41
GLA P06280 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
ATM Q13315 1/20 0.41
HSD17B10 Q99714 1/20 0.41
NPC1 O15118 1/20 0.40
PPARA Q07869 1/20 0.40
RAB9A P51151 1/20 0.40
POLB P06746 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11545452 0.86 USP2 (0.54) USP2ALDH1A1KDM4EGAAHPGD
SCHEMBL14879577 0.81 POLB (0.52) NOTUMALDH1A1HPGDMAPTPOLB
SCHEMBL14879713 0.78 RAB9A (0.50) USP2ALDH1A1KDM4EGAAHPGD
SCHEMBL14881379 0.78 KDM4E (0.56) USP2NOTUMALDH1A1KDM4EHPGD
SCHEMBL8075068 0.77 NOTUM (0.54) USP2NOTUMALDH1A1KDM4EGAA
SCHEMBL14879659 0.77 ALDH1A1 (0.51) USP2ALDH1A1KDM4EGAAHPGD
SCHEMBL2875469 0.77 HPGD (0.52) USP2ALDH1A1KDM4EGAAHPGD
SCHEMBL14879718 0.76 IDO1 (0.40) USP2NOTUMALDH1A1KDM4EHPGD
SCHEMBL27901095 0.76 NOTUM (0.51) USP2NOTUMALDH1A1KDM4EGAA
SCHEMBL11546125 0.76 POLB (0.55) USP2ALDH1A1HPGDMAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013059648-A1 2,3,5 TRISUBSTITUTED ARYL AND HETEROARYL AMINO DERIVATIVES, COMPOSITIONS, AND METHODS OF USE NEUROTHERAPEUTICS PHARMA, INC. (US) 2013-04-25 WO disclosed
WO-2013059648-A1 2,3,5 TRISUBSTITUTED ARYL AND HETEROARYL AMINO DERIVATIVES, COMPOSITIONS, AND METHODS OF USE NEUROTHERAPEUTICS PHARMA, INC. (US) 2013-04-25 WO disclosed