Chlorpheniramine

Chlorpheniramine

SCHEMBL14879822

CN(C)CCC(c1ccc(Cl)cc1)c1ccccn1.[CaH2]

nearest known ligand 0.97

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HRH1

The experimentally established mechanism targets of Chlorpheniramine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 known ✓ P35367 5/20 0.97
CHRM2 P08172 6/20 0.97
SLC6A2 P23975 6/20 0.97
SLC6A4 P31645 6/20 0.97
SLC6A3 Q01959 5/20 0.97
KCNH2 Q12809 5/20 0.97
HRH3 Q9Y5N1 5/20 0.97
CHRM1 P11229 4/20 0.97
ADRA2B P18089 4/20 0.97
HTR2A P28223 3/20 0.97
SCN1A P35498 3/20 0.97
SCN2A Q99250 3/20 0.97
SCN3A Q9NY46 3/20 0.97
CYP2D6 P10635 3/20 0.97
CHRM5 P08912 2/20 0.97
HRH2 P25021 2/20 0.97
NFKB1 P19838 2/20 0.97
THPO P40225 2/20 0.97
HTR2C P28335 2/20 0.97
TSHR P16473 2/20 0.97

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Chlorpheniramine SCHEMBL14879823 1.00 CHRM2 (0.97) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Chlorpheniramine SCHEMBL20956397 0.99 CHRM2 (1.00) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Chlorpheniramine SCHEMBL4220 0.99 CHRM2 (1.00) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Dexchlorpheniramine SCHEMBL3538 0.99 CHRM2 (1.00) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Chlorpheniramine SCHEMBL29687335 0.99 CHRM2 (1.00) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Chlorpheniramine SCHEMBL4314182 0.99 CHRM2 (1.00) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Chlorpheniramine SCHEMBL4219 0.99 CHRM2 (1.00) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Chlorpheniramine SCHEMBL5022351 0.97 CHRM2 (0.97) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Chlorpheniramine SCHEMBL506017 0.97 CHRM2 (0.97) CHRM2SLC6A2SLC6A4HRH1SLC6A3
Chlorpheniramine SCHEMBL10622596 0.97 CHRM2 (0.97) CHRM2SLC6A2SLC6A4HRH1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2694707-A1 MONOMERS CAPABLE OF DIMERIZING IN AN AQUEOUS SOLUTION, AND METHODS OF USING SAME Cornell University (US) 2014-02-12 EP disclosed
EP-2693883-A1 SILYL MONOMERS CAPABLE OF MULTIMERIZING IN AN AQUEOUS SOLUTION, AND METHODS OF USING SAME Cornell University (US) 2014-02-12 EP disclosed
WO-2013058824-A1 MONOMERS CAPABLE OF DIMERIZING IN AN AQUEOUS SOLUTION, AND METHODS OF USING SAME CORNELL UNIVERSITY (US) 2013-04-25 WO disclosed
WO-2013058825-A1 SILYL MONOMERS CAPABLE OF MULTIMERIZING IN AN AQUEOUS SOLUTION, AND METHODS OF USING SAME CORNELL UNIVERSITY (US) 2013-04-25 WO disclosed